Tamoxifen is a competitive inhibitor of peripheral estrogen receptor. And if earlier it was believed that the drug does not have the influence of estrogen, but today this view is totally rejected. In fact, the ratio of agonist and antagonist activity equal to 45/55. Tamoxifen is a chemically derived form triphenylethylene. The drug belongs to the group of sex hormones. Initially it was used for the treatment of cancer in women (breast cancer). But, undoubtedly, today Tamoxifen is much more common in sports and bodybuilding in particular.
It is no secret that the majority of steroids are exposed flavoring that is converted in to the female sex hormones – estrogens. This can lead to a variety of side effects, which is able to warn svoevremennyypriem Tamoxifen. Unlike other means such exposure, the substance is neither androgen or anabiotic.
- The increase in power performance.
- Increased hardness and muscle relief.
- The increase in muscle mass. Tamoxifen is very popular in bodybuilding Argued that without it can not do any one victory in major competitions.
- The marked anti-estrogen effects. The effect, which made so popular Tamoxifen. The higher dosage of AAC, the greater the need to compensate for estrogenic activity. Tamoxifen or analogues thereof at FCT after heavy courses practically mandatory.
- The fight against fat.
- Prevention of feminization.
- Reducing the risk of developing atherosclerosis, the prevention of cardiovascular disease.
- Improving liver.
Tamoxifen antiestrogen effects caused by blocking estrogen receptors (rather than the termination of the conversion of testosterone into estrogen, as many think). Preparation only freezes estrogenic activity, and does not prevent it entirely.
How to take Tamoxifen after the course
How to take Tamoxifen TamoksifenPriem after a course of steroids should be combined with an aromatase inhibitor, the most popular of which is Proviron (it is often used for the reason that it does not inhibit the production of growth hormone and inhibits aromatase, thereby increasing the concentration of anabolic hormones in the blood). Tamoxifen as a primary means of PCT is used in doses of 10 to 20 milligrams daily from the last week of the course and ending the second week of its completion. If Proviron is not accepted, Tamoxifen is included later – at 2 weeks, and ends 2-3 weeks after its cancellation.
Please note that the highest levels of estrogen in the body occurs at the end of the first week of the course AAS. As for how to take Tamoxifen bodybuilding on a course of steroids, flavoring has no effect, it is recommended to add it only at the end of the cycle.
The most common side effects of Tamoxifen associated with its pronounced antiestrogenic properties. Exceeding the recommended dose and / or duration of the course can cause female hair loss or total hair loss, flushing intense heat, itching, perineal pain in the bones; men – fever, dizziness, nausea. Because of the delay zhidkostimozhet disrupt the normal functioning of the kidneys. Also, sometimes there are bouts of depression, depression and drowsiness. Excessive intake is fraught with fatigue, constipation, and anorexia. You may experience inflammation of the retina, cataract, partial or complete loss of vision. Tamoxifen is sometimes accompanied by a rash on the skin. Cases of headache, changes in the cornea, unclear consciousness. Liver occur only in case of serious diseases of the body (such as hepatitis).
Reviews of Tamoxifen
Reviews often expressed about the preparation of the athletes not as Tamoxifen for many years been used in post-menopausal women with estrogen-receptor-positive, and breast cancer patients. As for athletes, they are a marked anti-estrogen effects. Despite the wide range of possible side effects of Tamoxifen reviews indicate that adverse reactions are extremely rare.
Women athletes talk about the impossibility of use of the drug during pregnancy. In addition, it can prevent the implantation of the egg in the uterine wall. Reviews of tamoxifen on entry-level athletes are rare because amateurs are often bypassed by simple solo AAS courses that do not require FCT.